A new synthetic route of 3034-38-6

According to the analysis of related databases, 3034-38-6, the application of this compound in the production field has become more and more popular.

Each compound has different characteristics, and only by selecting the characteristics of the compound suitable for a specific situation can the compound be applied on a large scale. 3034-38-6, name is 5-Nitro-1H-imidazole, This compound has unique chemical properties. The synthetic route is as follows., Product Details of 3034-38-6

General procedure: The opportune alkyl bromide (916 mg, 4.26 mmol) was added to a solution of 4-nitro-1H-imidazole5 (438 mg, 3.87 mmol) in acetonitrile (3 mL) and potassium carbonate (803 mg, 5.81 mmol).The resulting mixture was heated at 60 C overnight. The reaction mixture was then filtered, andthe filtrate was concentrated in vacuum, leaving a yellow solid. The desired product was recoveredfrom this residue by normal phase column chromatography on a cartridge Biotage HP-SiO2 (50 g)column primed with DCM only. The column was then run for 4CV with DCM and then changed toDCM/MeOH 9:1 over 5CV.1-[2-(2-Methoxyphenyl)ethyl]-4-nitro-1H-imidazole (6a): White solid, 82% yield, mp: 100-102 C; IR: nu= 1338 (NO) cm-1; 1H NMR (400 MHz, DMSO-d6) delta = ppm 3.11 (t, J = 7.34 Hz, 2H), 3.75 (s, 3H), 4.28(t, J = 7.34 Hz, 2H), 6.84 (t, J = 7.34 Hz, 1H) 6.93-7.06 (m, 2H), 7.19-7.26 (m, 1H), 7.67 (s, 1H), 8.30 (s, 1H); 13C NMR (100 MHz, DMSO-d6) delta = ppm 158.8, 146.2, 138.7, 129.9, 128.4, 126.8, 121.5, 120.4, 112.9,56.8, 49.6, 28.6; HRMS (ESI): m/z calcd. for C12H13N3O3 248.9567 [M + H]+, found 248.9542.

According to the analysis of related databases, 3034-38-6, the application of this compound in the production field has become more and more popular.

Reference:
Article; Francini, Cinzia Maria; Musumeci, Francesca; Fallacara, Anna Lucia; Botta, Lorenzo; Molinari, Alessio; Artusi, Roberto; Mennuni, Laura; Angelucci, Adriano; Schenone, Silvia; Molecules; vol. 23; 9; (2018);,
Imidazole – Wikipedia,
Imidazole | C3H4N2 – PubChem